UniProt O94804
O94804
O94804 (UniProt O94804): 24 experimental structures on GenesisL1, 8 ligands bound. Binding sites, pockets, druggability and 3D structures in GL1X.
- UniProt
- O94804
- Experimental structures
- 24
- Predicted models
- 0
- Ligands
- 8
Structures
24 records of O94804 in the MolNFT archive: 24 experimental, 0 predicted.
| Entry | Title | Method | Chains | Ligands | Pockets |
|---|---|---|---|---|---|
| 2J7T | Crystal structure of human serine threonine kinase-10 bound to SU11274 | x-ray diffraction | A | — | — |
| 2J7T | Crystal structure of human serine threonine kinase-10 bound to SU11274 | x-ray diffraction | A | — | — |
| 4AOT | Crystal Structure of Human Serine Threonine Kinase-10 (LOK) Bound to GW830263A | x-ray diffraction | A, B | — | — |
| 4AOT | Crystal structure of human serine threonine kinase-10 (lok) bound to GW830263A | x-ray diffraction | A, B | — | — |
| 4BC6 | Crystal structure of human serine threonine kinase-10 bound to novel Bosutinib Isoform 1… | x-ray diffraction | A | — | — |
| 4BC6 | Crystal structure of human serine threonine kinase-10 bound to novel bosutinib isoform 1… | x-ray diffraction | A | — | — |
| 4EQU | Human STK-10 (LOK) kinase domain in DFG-out conformation with inhibitor DSA-7 | x-ray diffraction | A, B | — | — |
| 4EQU | Human stk-10 (lok) kinase domain in dfg-out conformation with inhibitor dsa-7 | x-ray diffraction | A, B | — | — |
| 4USD | Human STK10 (LOK) with SB-633825 | x-ray diffraction | A, B | — | — |
| 4USD | Human STK10 (lok) with sb-633825 | x-ray diffraction | A, B | — | — |
| 4USE | Human STK10 (LOK) with SB-633825 | x-ray diffraction | A, B | — | — |
| 4USE | Human STK10 (lok) with sb-633825 | x-ray diffraction | A, B | — | — |
| 5AJQ | Human LOK (STK10) in complex with Bosutinib | x-ray diffraction | A, B | — | — |
| 5AJQ | Human lok (STK10) in complex with bosutinib | x-ray diffraction | A, B | — | — |
| 5OWQ | Human STK10 bound to dovitinib | x-ray diffraction | A, B | 38O | — |
| 5OWR | Human STK10 bound to dasatinib | x-ray diffraction | A | 1N1 | — |
| 6EIM | Human STK10 bound to GW683134A | x-ray diffraction | A, B | B6E | — |
| 6EIM | Human STK10 bound to GW683134A | x-ray diffraction | A, B | B6E | — |
| 6GTT | Human STK10 bound to birb-796 | x-ray diffraction | A | B96 | — |
| 6HXF | Human STK10 bound to a maleimide inhibitor | x-ray diffraction | B, A, C, D | R70, CL | — |
| 6HXF | Human STK10 bound to a maleimide inhibitor | x-ray diffraction | B, A, C, D | R70, CL | — |
| 6I2Y | Human STK10 bound to foretinib | x-ray diffraction | A, B | 88Z | — |
| 7QGP | STK10 (lok) bound to macrocycle CKJB51 | x-ray diffraction | A | DJ8, CL | — |
| O94804 | AlphaFold monomer V2.0 prediction for SERINE/THREONINE-protein kinase 10 (O94804) | — | — | — |
Ligands
- CL · Chloride ion · in 3 records
- B6E · ~{N}-[5-[4-[[2-fluoranyl-5-(trifluoromethyl) phenyl]carbamoylamino]phenoxy]-1~{H}-benzimidazol-2-yl]furan-2-carboxamide · in 2 records
- R70 · 3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl) phenyl]amino]pyrrole-2,5-dione · in 2 records
- 1N1 · N-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide · in 1 record
- 38O · 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]quinolin-2(1H)-one · in 1 record
- 88Z · N-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy) quinolin-4-yl]oxy}phenyl)-N'-(4-fluorophenyl) cyclopropane-1,1-dicarboxamide · in 1 record
- B96 · 1-(5-tert-butyl-2-P-tolyl-2H-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea · in 1 record
- DJ8 · 1-[(4-chloranyl-2-methyl-phenyl)methyl]-3-(7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17, 20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaen-5-yl) urea · in 1 record
Elsewhere
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