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UniProt Q59957

DNA gyrase subunit B (Q59957)

DNA gyrase subunit B (UniProt Q59957), EC 5.99.1.3: 6 experimental structures on GenesisL1, 3 ligands bound, 40 pockets. Binding sites, pockets, druggability and 3D structures in GL1X.

UniProt
Q59957
Protein
DNA gyrase subunit B
EC
5.99.1.3
Experimental structures
6
Predicted models
0
Ligands
3
Pockets
40 · 3 records with a druggable one

Structures

6 records of Q59957 in the MolNFT archive: 6 experimental, 0 predicted.

EntryTitleMethodChainsLigandsPockets
4Z2CQuinolone(Moxifloxacin)-DNA cleavage complex of gyrase from S. pneumoniaex-ray diffractionC, DMFX13 (best 0.83)
4Z2CQUINOLONE(MOXIFLOXACIN)-DNA cleavage complex of gyrase from S. pneumoniaex-ray diffractionC, D——
4Z2DQuinolone(Levofloxacin)-DNA cleavage complex of gyrase from S. pneumoniaex-ray diffractionC, DLFX12 (best 0.74)
4Z2DQUINOLONE(LEVOFLOXACIN)-DNA cleavage complex of gyrase from S. pneumoniaex-ray diffractionC, D——
4Z2EQuinolone(Trovafloxacin)-DNA cleavage complex of gyrase from S. pneumoniaex-ray diffractionC, DTR615 (best 0.78)
4Z2EQUINOLONE(TROVAFLOXACIN)-DNA cleavage complex of gyrase from S. pneumoniaex-ray diffractionC, D——

Ligands

  • LFX · (3S)-9-fluoro-3-methyl-10-(4-methylpiperazin-1-yl)-7-oxo-2,3-dihydro-7H-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxylic acid · in 1 record
  • MFX · 1-cyclopropyl-6-fluoro-8-methoxy-7-[(4aS,7aS)-octahydro-6H-pyrrolo[3,4-b]pyridin-6-yl]-4-oxo-1,4-dihydroquinoline-3-carboxylic acid · in 1 record
  • TR6 · Trovafloxacin · in 1 record

Elsewhere

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