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UniProt G5E8H1

Glutamate receptor (G5E8H1)

Glutamate receptor (UniProt G5E8H1): 4 experimental structures on GenesisL1, 6 ligands bound, 18 pockets. Binding sites, pockets, druggability and 3D structures in GL1X.

UniProt
G5E8H1
Protein
Glutamate receptor
Experimental structures
4
Predicted models
0
Ligands
6
Pockets
18 · 2 records with a druggable one

Structures

4 records of G5E8H1 in the MolNFT archive: 4 experimental, 0 predicted.

EntryTitleMethodChainsLigandsPockets
7LDDnative AMPA receptorelectron microscopyB, DNAG, D10, ZK1, D12, C14, HP69 (best 0.83)
7LDDNative AMPA receptorelectron microscopyB, DNAG, ZK1, D12, C14—
7LDEnative AMPA receptorelectron microscopyB, DNAG, D10, ZK1, D12, C14, HP69 (best 0.83)
7LDENative AMPA receptorelectron microscopyB, DNAG, ZK1, D12, C14—

Ligands

  • C14 · Tetradecane · in 4 records
  • D12 · Dodecane · in 4 records
  • NAG · 2-acetamido-2-deoxy-beta-D-glucopyranose · in 4 records
  • ZK1 · {[7-morpholin-4-yl-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl]methyl}phosphonic acid · in 4 records
  • D10 · Decane · in 2 records
  • HP6 · Heptane · in 2 records

Elsewhere

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