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UniProt A5U9I4

TetR-family transcriptional regulatory repressor protein (A5U9I4)

TetR-family transcriptional regulatory repressor protein (UniProt A5U9I4): 8 experimental structures on GenesisL1, 5 ligands bound, 1 pocket. Binding sites, pockets, druggability and 3D structures in GL1X.

UniProt
A5U9I4
Protein
TetR-family transcriptional regulatory repressor protein
Experimental structures
8
Predicted models
0
Ligands
5
Pockets
1 · 1 record with a druggable one

Structures

8 records of A5U9I4 in the MolNFT archive: 8 experimental, 0 predicted.

EntryTitleMethodChainsLigandsPockets
5IOYStructure of Transcriptional Regulatory Repressor Protein - EthR from Mycobacterium Tuberculosis in…x-ray diffractionA6C5, SO4—
5IOYStructure of transcriptional regulatory repressor protein - ethr from mycobacterium tuberculosis in…x-ray diffractionA——
5IOZStructure of Transcriptional Regulatory Repressor Protein - EthR from Mycobacterium Tuberculosis in…x-ray diffractionA6C4—
5IOZStructure of transcriptional regulatory repressor protein - ethr from mycobacterium tuberculosis in…x-ray diffractionA——
5IP6Structure of Transcriptional Regulatory Repressor Protein - EthR from Mycobacterium Tuberculosis in…x-ray diffractionA6C9—
5IP6Structure of transcriptional regulatory repressor protein - ethr from mycobacterium tuberculosis in…x-ray diffractionA——
5IPAStructure of Transcriptional Regulatory Repressor Protein - EthR from Mycobacterium Tuberculosis in…x-ray diffractionA6C81 (best 0.75)
5IPAStructure of transcriptional regulatory repressor protein - ethr from mycobacterium tuberculosis in…x-ray diffractionA——

Ligands

  • 6C4 · N-(cyclopentylmethyl)cyclopentanecarboxamide · in 1 record
  • 6C5 · N-(cyclopentylmethyl)pyrrolidine-1-carboxamide · in 1 record
  • 6C8 · (2E)-3-(furan-3-yl)-1-(pyrrolidin-1-yl)prop-2-en-1-one · in 1 record
  • 6C9 · N-{[(3S)-oxolan-3-yl]methyl}pyrrolidine-1-carboxamide · in 1 record
  • SO4 · Sulfate ion · in 1 record

Elsewhere

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