GL1X · GenesisL1 explorer

MolNFT v1 · #94472 · protein

BRD4 bromodomain 1 complex with N-[3-(2-oxo-2,3-dihydro-1,3-thiazol-4- YL)PHENYL]THIOPHENE-2-sulfonamide inhibitor

4HXR: “BRD4 bromodomain 1 complex with N-[3-(2-oxo-2,3-dihydro-1,3-thiazol-4- YL)PHENYL]THIOPHENE-2-sulfonamide…”. X-ray diffraction. MolNFT v1 #94472 on GenesisL1: 3D structure, binding sites and pockets in GL1X.

PDB
4HXR
Type
protein
Length
125 residues
Chains
1
Method
x-ray diffraction
Collection
MolNFT v1 / PDB
Contract
0xDE3723766Bc32dcACD03C17BaA400A7B36837Eba
Owner
0x3396CDB397284571d12822B4ae1189a8E22AAAAA
UniProt
O60885

Structure

x-ray diffraction · 1 distinct chain.

ChainMoleculeTypeResiduesSecondary structureUniProt
A—protein125—O60885

Compared structures

  • 4HXR · Brd4 Bromodomain 1 complex with N-[3-(2-OXO-2,3-DIHYDRO-1,3-THIAZOL-4-YL)PHENYL]THIOPHENE… · the same entry in another collection · chain A against A, TM-score 1.00
  • O60885 · AlphaFold monomer V2.0 prediction for bromodomain-containing protein 4 (O60885) · a predicted model of the same protein · chain A against A, TM-score 0.97

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