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UniProt U3KMH2

Transcription initiation factor TFIID subunit (U3KMH2)

Transcription initiation factor TFIID subunit (UniProt U3KMH2): 3 experimental structures on GenesisL1, 2 ligands bound, 4 pockets. Binding sites, pockets, druggability and 3D structures in GL1X.

UniProt
U3KMH2
Protein
Transcription initiation factor TFIID subunit
Experimental structures
3
Predicted models
0
Ligands
2
Pockets
4 · 1 record with a druggable one

Structures

3 records of U3KMH2 in the MolNFT archive: 3 experimental, 0 predicted.

EntryTitleMethodChainsLigandsPockets
6DF4TAF1-BD2 in complex with CPD8 (6-(but-3-en-1-yl)-4-(3-(morpholine-4…x-ray diffractionAG9Y—
6DF7TAF1-BD2 in complex with Cpd27 (6-(but-3-en-1-yl)-4-(1-methyl-6-(morpholine-4-carbonyl)-1H-benzo[d]i…x-ray diffractionA, BG9V4 (best 0.65)
6DF7TAF1-BD2 in complex with CPD27 (6-(but-3-en-1-yl)-4-(1-methyl-6…x-ray diffractionA, BG9V—

Ligands

  • G9V · 6-(but-3-en-1-yl)-4-[1-methyl-6-(morpholine-4-carbonyl)-1H-benzimidazol-4-yl]-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one · in 2 records
  • G9Y · 6-(but-3-en-1-yl)-4-[3-(morpholine-4-carbonyl)phenyl]-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one · in 1 record

Elsewhere

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