UniProt Q9XB24
Beta-lactamase (Q9XB24)
Beta-lactamase (UniProt Q9XB24), EC 3.5.2.6: 14 experimental structures on GenesisL1, 5 ligands bound, 4 pockets. Binding sites, pockets, druggability and 3D structures in GL1X.
- UniProt
- Q9XB24
- Protein
- Beta-lactamase
- EC
- 3.5.2.6
- Experimental structures
- 14
- Predicted models
- 0
- Ligands
- 5
- Pockets
- 4 · 3 records with a druggable one
Structures
14 records of Q9XB24 in the MolNFT archive: 14 experimental, 0 predicted.
| Entry | Title | Method | Chains | Ligands | Pockets |
|---|---|---|---|---|---|
| 6K8X | Crystal structure of a class C beta lactamase | x-ray diffraction | A | — | — |
| 6K8X | Crystal structure of a class C beta lactamase | x-ray diffraction | A | — | — |
| 6K9T | Crystal structure of a class C beta-lactamase in complex with cefotaxime | x-ray diffraction | A | CEF | — |
| 6K9T | Crystal structure of a class C beta-lactamase in complex with cefotaxime | x-ray diffraction | A | CEF | — |
| 6KA5 | Crystal structure of a class C beta-lactamase in complex with cefoxitin | x-ray diffraction | A | 1S7 | — |
| 6KA5 | Crystal structure of a class C beta-lactamase in complex with cefoxitin | x-ray diffraction | A | 1S7 | — |
| 6KBY | Crystal structure of a class C beta lactamase in complex with AMP | x-ray diffraction | A | AMP | 2 (best 0.62) |
| 6KBY | Crystal structure of a class C beta lactamase in complex with AMP | x-ray diffraction | A | AMP | — |
| 6M5H | A class C beta-lactamase mutant - Y150F | x-ray diffraction | A | — | — |
| 6M5H | A class C beta-lactamase mutant - Y150F | x-ray diffraction | A | — | — |
| 6M5P | A class C beta-lactamase | x-ray diffraction | A | MER | 1 (best 0.53) |
| 6M5P | A class C beta-lactamase | x-ray diffraction | A | MER | — |
| 6M5Q | A class C beta-lactamase mutant - Y150F | x-ray diffraction | A | IM2 | 1 (best 0.54) |
| 6M5Q | A class C beta-lactamase mutant - Y150F | x-ray diffraction | A | IM2 | — |
Ligands
- 1S7 · (2R)-2-{(1S)-1-methoxy-2-oxo-1-[(thiophen-2-ylacetyl) amino]ethyl}-5-methylidene-5,6-dihydro-2H-1,3-thiazine-4-carboxylic acid · in 2 records
- AMP · Adenosine monophosphate · in 2 records
- CEF · CEFOTAXIME, C3' cleaved, open, bound form · in 2 records
- IM2 · (5R)-5-[(1S,2R)-1-formyl-2-hydroxypropyl]-3-[(2-{[(E)-iminomethyl]amino}ethyl)sulfanyl]-4,5-dihydro-1H-pyrrole-2-carbox ylic acid · in 2 records
- MER · (4R,5S)-3-{[(3S,5S)-5-(dimethylcarbamoyl)pyrrolidin-3-yl]sulfanyl}-5-[(2S,3R)-3-hydroxy-1-oxobutan-2-yl]-4-methyl-4,5-dihydro-1H-pyrrole-2-carboxylic acid · in 2 records
Elsewhere
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