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UniProt Q7KZI7

Q7KZI7

Q7KZI7 (UniProt Q7KZI7): 7 experimental structures on GenesisL1, 3 ligands bound. Binding sites, pockets, druggability and 3D structures in GL1X.

UniProt
Q7KZI7
Experimental structures
7
Predicted models
0
Ligands
3

Structures

7 records of Q7KZI7 in the MolNFT archive: 7 experimental, 0 predicted.

EntryTitleMethodChainsLigandsPockets
3IECHelicobacter pylori CagA Inhibits PAR1/MARK Family Kinases by Mimicking Host Substratesx-ray diffractionA, B, C, D——
3IECHelicobacter pylori caga inhibits PAR1/MARK family kinases by mimicking host substratesx-ray diffractionA, B, C, D——
5EAKOptimization of Microtubule Affinity Regulating Kinase (MARK) Inhibitors with Improved Physical…x-ray diffractionA, B24R—
5EAKOptimization of microtubule affinity regulating kinase (mark) inhibitors with improved physical…x-ray diffractionA, B——
5KZ7MARK2 complex with 7-[(1S)-1-(4-FLUOROPHENYL)ETHYL]-5,5-dimethyl-2-(3…x-ray diffractionA, B6Z2—
5KZ8MARK2 complex with 7-[(1S)-1-(4-FLUOROPHENYL)ETHYL]-5,5-dimethyl-2-(3…x-ray diffractionA, B6Z5—
Q7KZI7AlphaFold monomer V2.0 prediction for SERINE/THREONINE-protein kinase MARK2 (Q7KZI7)———

Ligands

  • 24R · N-[(1S,2R)-2-aminocyclohexyl]-4-[6-(1-methyl-1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamide · in 1 record
  • 6Z2 · 7-[(1~{S})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-one · in 1 record
  • 6Z5 · 5,5-dimethyl-7-[(1~{S})-4-oxidanyl-1~{H}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-one · in 1 record

Elsewhere

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