GL1X · GenesisL1 explorer

UniProt A0A4V5JMQ9

DNA gyrase subunit B (A0A4V5JMQ9)

DNA gyrase subunit B (UniProt A0A4V5JMQ9), EC 5.6.2.2: 8 experimental structures on GenesisL1, 4 ligands bound, 6 pockets. Binding sites, pockets, druggability and 3D structures in GL1X.

UniProt
A0A4V5JMQ9
Protein
DNA gyrase subunit B
EC
5.6.2.2
Experimental structures
8
Predicted models
0
Ligands
4
Pockets
6 · 3 records with a druggable one

Structures

8 records of A0A4V5JMQ9 in the MolNFT archive: 8 experimental, 0 predicted.

EntryTitleMethodChainsLigandsPockets
6KZVCrystal structure of E.coli DNA gyrase B in complex with 2-oxo-1,2-dihydroquinoline derivativex-ray diffractionAE0F2 (best 0.54)
6KZVCrystal structure of E.COLI DNA gyrase B in complex with 2-oxo-1,2- dihydroquinoline derivativex-ray diffractionAE0F—
6KZXCrystal structure of E.coli DNA gyrase B in complex with 2-oxo-1,2-dihydroquinoline derivativex-ray diffractionAE0L—
6KZXCrystal structure of E.COLI DNA gyrase B in complex with 2-oxo-1,2- dihydroquinoline derivativex-ray diffractionAE0L—
6KZZCrystal structure of E.coli DNA gyrase B in complex with 2-oxo-1,2-dihydroquinoline derivativex-ray diffractionAE0R2 (best 0.51)
6KZZCrystal structure of E.COLI DNA gyrase B in complex with 2-oxo-1,2- dihydroquinoline derivativex-ray diffractionAE0R—
6L01Crystal structure of E.coli DNA gyrase B in complex with 2-oxo-1,2-dihydroquinoline derivativex-ray diffractionAE0U2 (best 0.52)
6L01Crystal structure of E.COLI DNA gyrase B in complex with 2-oxo-1,2- dihydroquinoline derivativex-ray diffractionAE0U—

Ligands

  • E0F · ~{N}-[2-[[cyclohexyl(methyl)amino]methyl]phenyl]-2-oxidanylidene-1~{H}-quinoline-3-carboxamide · in 2 records
  • E0L · 3-[[8-(methylamino)-2-oxidanylidene-1~{H}-quinolin-3-yl]carbonylamino]benzoic acid · in 2 records
  • E0R · 4-[[8-(methylamino)-2-oxidanylidene-1~{H}-quinolin-3-yl]carbonylamino]benzoic acid · in 2 records
  • E0U · 2-[3-[[8-(methylamino)-2-oxidanylidene-1~{H}-quinolin-3-yl]carbonylamino]phenyl]ethanoic acid · in 2 records

Elsewhere

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