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UniProt A0A045KCS8

EthR (A0A045KCS8)

EthR (UniProt A0A045KCS8): 8 experimental structures on GenesisL1, 4 ligands bound, 1 pocket. Binding sites, pockets, druggability and 3D structures in GL1X.

UniProt
A0A045KCS8
Protein
EthR
Experimental structures
8
Predicted models
0
Ligands
4
Pockets
1 · 1 record with a druggable one

Structures

8 records of A0A045KCS8 in the MolNFT archive: 8 experimental, 0 predicted.

EntryTitleMethodChainsLigandsPockets
5EYRStructure of Transcriptional Regulatory Repressor Protein - EthR from Mycobacterium Tuberculosis in…x-ray diffractionA5T0—
5EYRStructure of transcriptional regulatory repressor protein - ethr from mycobacterium tuberculosis in…x-ray diffractionA——
5J1RStructure of Transcriptional Regulatory Repressor Protein - EthR from Mycobacterium Tuberculosis in…x-ray diffractionA6FG—
5J1RStructure of transcriptional regulatory repressor protein - ethr from mycobacterium tuberculosis in…x-ray diffractionA——
5J1UStructure of Transcriptional Regulatory Repressor Protein - EthR from Mycobacterium Tuberculosis in…x-ray diffractionAP93—
5J1UStructure of transcriptional regulatory repressor protein - ethr from mycobacterium tuberculosis in…x-ray diffractionA——
5J1YStructure of Transcriptional Regulatory Repressor Protein - EthR from Mycobacterium Tuberculosis in…x-ray diffractionAP871 (best 0.72)
5J1YStructure of transcriptional regulatory repressor protein - ethr from mycobacterium tuberculosis in…x-ray diffractionA——

Ligands

  • 5T0 · 3-[1-[4-(methylaminomethyl)phenyl]piperidin-4-yl]-1-pyrrolidin-1-yl-propan-1-one · in 1 record
  • 6FG · 3-(furan-3-yl)-1-(pyrrolidin-1-yl)propan-1-one · in 1 record
  • P87 · 3-[(3S)-oxolan-3-yl]-1-(pyrrolidin-1-yl)propan-1-one · in 1 record
  • P93 · N-[(furan-3-yl)methyl]pyrrolidine-1-carboxamide · in 1 record

Elsewhere

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