Ligand · 8KH
8KH · N-[5-[4-[[5-[[(2S)-3,3-dimethyl-1-[(2S,4R)-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]-4-oxidanyl-pyrrolidin-1-yl]-1-oxidanylidene-butan-2-yl]amino]-5-oxidanylidene-pentyl]carbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl]-6-oxidanylidene-4-(trifluoromethyl)-1H-pyridine-3-carboxamide
8KH, N-[5-[4-[[5-[[(2S)-3,3-dimethyl-1-[(2S,4R)-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]-4-oxidanyl-pyrrolidin-1-yl]-1-oxidanylidene-butan-2-yl]amino]-5-oxidanylidene-pentyl]carbamoyl]phenyl]-2-(4-methylpiperazin-1-yl)phenyl…
- Component
- 8KH
- Formula
- C52 H60 F3 N9 O7 S
- Class
- ligand
- Structures
- 1
- PDB entries
- 1
Binding sites
8KH in 1 structure; the first of them:
- 7Q2J · Quaternary complex of human WDR5 and PVHL:ELONGINC:ELONGINB bound to protac homer · 8KH D401 · binds ASN67, PHE76, PRO86, TRP88, PHE91, TYR98, PRO99, LEU101 and 23 more
Residues it binds most
PHE 1, SER 1, ILE 1, TYR 1, ASP 1, HIS 1, LEU 1, PRO 1, TRP 1, ALA 1 (residue and the binding sites it lines).
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